付建国

发布者:创新中药1发布时间:2021-04-25浏览次数:1074

姓名:付建国性别:
职称:副研究员学历:博士研究生
专家类别:硕士生导师职务:创新中药研究院团支部书记
电话:
传真:
电子邮箱:

fujg@shutcm.edu.cn

通讯地址:蔡伦路1200号
个人主页:

招生专业:

院系名称专业大类一级学科专业代码/专业名称学位类型招生类型
创新中药研究院理学中药学100800/中药学学术型硕士

个人简历:

2023.01-目前
副研究员,上海中医药大学 创新中药研究院 手性药物研究中心
2020.07-2022.12助理研究员,上海中医药大学 创新中药研究院 手性药物研究中心
2018.03-2020.06师资博士后,上海中医药大学 中药学专业 合作导师:林国强 研究员
2011.09-2016.07博士,中国科学院上海有机化学研究所,有机化学专业(导师:林国强 研究员)
2007.09-2011.07本科,吉林大学化学学院,化学专业(导师:寮渭巍 教授)

研究内容:

中药活性分子的合成与修饰
药物化学

主持科研项目:

课题名称项目名称起止时间金额
生物活性导向的Lycodine型石松生物碱的多样性合成研究国家自然科学基金青年项目2024.01-2026.1230万

非介导型钯催化芳基卤代物串联双偶联反应研究

上海市“科技行动计划”自然科学基金面上项目

2022.04-2025.0320万

基于靶向抑制Lyn/FcεRIβ的新型抗过敏药物的研究

上海中医药大学预算内科研项目

2021.11-2023.01

5万

发表文章:

1. Jun-Jie Wang; Rui-Xue Bai; Mao-Qi Yang; Zheng-Yu Chen; Min-Dan Wang; Qian Zhao*; Guo-Qiang Lin; Jian-Guo Fu*; Chen-Guo Feng*, Total Synthesis of (-)-Amathaspiramide A via One-pot Aldol Addition/Transamidification Reaction. Organic Chemistry Frontiers. 2022, 9(11), 3045-3049. (IF = 5.456)

2Ze-Jian Xue; Han-Yu Lu; Jian-Guo Fu*; Chen-Guo Feng*; Guo-Qiang Lin*An azo-bridged ring system enabled by-standing immobilization of a chiral diene ligand, Organic Chemistry Frontiers, 2021, 8(19), 5397-5402.(IF = 5.456)

3. Xiao-Ming Ji; Yan-Zhen Chen; Jian-Guo Fu*; Shu-Sheng Zhang; Chen-Guo Feng*, Phosphorylation of C(sp3)–H Bonds via 1,4-Palladium Migration. Organic Letters, 2022, 24(21): 3781-3785. (IF = 6.072)

4Yi-Kang Song; Si-Yu Xu; Shu-Sheng Zhang; Jian-Guo Fu*; Guo-Qiang Lin; Chen-Guo Feng*, Palladium-Catalyzed Tandem γ-Arylation/Aromatization of Cyclohex-2-En-1-One Derivatives: A Route to 3,4- Dihydroanthracen-1(2H)-One,Advanced Synthesis & Catalysis, 2021, 363(12): 3001-3005. (IF = 5.981)

5. Yi-Kang Song#, Li Liu#, Jun-Jie Wang, Fei Qian, Mao-Qi Yang, Liu-Qiang Zhang*, Jian-Guo Fu*, Yi-Ming Li, Chen-Guo Feng*, An Asymmetric Synthesis of (+)-Scrodentoid A from Dehydroabietic Acid, Tetrahedron, 2021, 85, 132031. (IF = 2.388)

6. Shao-Dong Lv, Tian Tian, Liu-Qiang Zhang, Si-Yu Xu, Dong-Hai Zhao, Jun-Jie Wang, Jian-Guo Fu*, Yi-Ming Li*, Chen-Guo Feng*, Total synthesis of (±)-Scrodentoid A, Tetrahedron, 2019, 75(52): 130774. (IF = 2.388)

7. Jian-Guo Fu, Guang-Qiang Xu, Rui Ding, Guo-Qiang Lin, Bing-Feng Sun*, Asymmetric Total Synthesis of Lycopodium Alkaloids α-Obscurine, N-desmethyl-α-Obscurine, β-Obscurine and N-desmethyl-β-Obscurine, Organic Chemistry Frontiers, 2016, 3(1): 62-65.(IF = 5.456)

8. Jian-Guo Fu#, Yi-Fan Shan#, Wang-Bin Sun, Guo-Qiang Lin, Bing-Feng Sun*, An Asymmetric Approach to Bicyclo[2.2.1]heptane-1-carboxylates via a Formal [4+2] Cycloaddition Reaction Enabled by Organocatalysis, Organic & Biomolecular Chemistry, 2016, 14(23): 5229-5232. (IF = 3.89)

9. Rui Ding#Jian-Guo Fu#, Guang-Qiang Xu, Bing-Feng Sun*, Guo-Qiang Lin*, Divergent Total Synthesis of the Lycopodium Alkaloids Huperzine A, Huperzine B, and Huperzine U, The Journal of Organic Chemistry, 2014, 79(1): 240-250. (IF = 4.198)

10. Jian-Guo Fu, Rui Ding, Bing-Feng Sun*, Guo-Qiang Lin*, Wagner-Meerwein Rearrangement of [3.3.1] Bicyclic N-Boc Aminols: Vinyl Migration in preference to Aryl Migration, Tetrahedron, 2014, 70(44): 8374-8379. (IF = 2.388)